BIOMEMBRANAS
BIOMEMBRANAS
Università di Perugia
Perugia, ItaliaPublications in collaboration with researchers from Università di Perugia (11)
2023
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New bioisosteric sulphur-containing choline kinase inhibitors with a tracked mode of action
European journal of medicinal chemistry, Vol. 246, pp. 115003
2022
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Anticancer Activity of the Choline Kinase Inhibitor PL48 Is Due to Selective Disruption of Choline Metabolism and Transport Systems in Cancer Cell Lines
Pharmaceutics, Vol. 14, Núm. 2
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Biological Evaluation of New Thienopyridinium and Thienopyrimidinium Derivatives as Human Choline Kinase Inhibitors
Pharmaceutics, Vol. 14, Núm. 4
2021
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3-hydroxy-L-kynurenamine is an immunomodulatory biogenic amine
Nature Communications, Vol. 12, Núm. 1
2020
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Flow synthesis of biologically-relevant compound libraries
Molecules, Vol. 25, Núm. 4
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Synthesis, biological evaluation, in silico modeling and crystallization of novel small monocationic molecules with potent antiproliferative activity by dual mechanism
European Journal of Medicinal Chemistry, Vol. 207
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Targeting Aryl hydrocarbon receptor for next-generation immunotherapies: Selective modulators (SAhRMs) versus rapidly metabolized ligands (RMAhRLs)
European Journal of Medicinal Chemistry, Vol. 185
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Waste minimized synthesis of pharmaceutically active compounds: Via heterogeneous manganese catalysed C-H oxidation in flow
Green Chemistry, Vol. 22, Núm. 2, pp. 397-403
2018
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Lead optimization-hit expansion of new asymmetrical pyridinium/quinolinium compounds as choline kinase α1 inhibitors
Future Medicinal Chemistry, Vol. 10, Núm. 15, pp. 1769-1786
2015
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Pharmacophore-Based Virtual Screening to Discover New Active Compounds for Human Choline Kinase α1
Molecular Informatics, Vol. 34, Núm. 6-7, pp. 458-466
2014
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Choline kinase active site provides features for designing versatile inhibitors
Current Topics in Medicinal Chemistry, Vol. 14, Núm. 23, pp. 2684-2693