ANA
CONEJO GARCÍA
CATEDRÁTICA DE UNIVERSIDAD
Publicaciones en las que colabora con ANA CONEJO GARCÍA (24)
2024
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Hydroxytyrosyl punicate: A first overview of a novel phenolipid with antiproliferative and antitrypanosomal activity
Journal of Functional Foods, Vol. 117
2023
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N-aryltetrahydroisoquinoline derivatives as HA-CD44 interaction inhibitors: Design, synthesis, computational studies, and antitumor effect
European Journal of Medicinal Chemistry, Vol. 258
2022
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Selective Anticancer Therapy Based on a HA-CD44 Interaction Inhibitor Loaded on Polymeric Nanoparticles
Pharmaceutics, Vol. 14, Núm. 4
2021
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Recent advances in the design of choline kinase α inhibitors and the molecular basis of their inhibition
Medicinal Research Reviews, Vol. 41, Núm. 2, pp. 902-927
2017
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Choline kinase inhibition and docking studies of a series of 6-(benzylthio)-9H-purin-9-yl-pyridinium derivatives
Medicinal Chemistry Research, Vol. 26, Núm. 11, pp. 2809-2815
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Lysophosphatidylcholine Regulates Sexual Stage Differentiation in the Human Malaria Parasite Plasmodium falciparum
Cell, Vol. 171, Núm. 7, pp. 1532-1544.e15
2016
2014
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Discovery of a new binding site on human choline kinase α1: Design, synthesis, crystallographic studies, and biological evaluation of asymmetrical bispyridinium derivatives
Journal of Medicinal Chemistry, Vol. 57, Núm. 2, pp. 507-515
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In vitro antiplasmodial and cytotoxic activities of asymmetrical pyridinium derivatives
European Journal of Medicinal Chemistry, Vol. 85, pp. 289-292
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NMR spectroscopic characterization of new nonsymmetrical bispyridinium choline kinase inhibitors
Magnetic Resonance in Chemistry
2013
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Antiproliferative activity, cell cycle, and apoptosis studies of a series of 6-substituted 9H-purin-9-yl-pyridinium derivatives on a human cervical carcinoma cell line
ChemMedChem, Vol. 8, Núm. 8, pp. 1266-1269
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Determination of potential scaffolds for human choline kinase α1 by chemical deconvolution studies
ChemBioChem, Vol. 14, Núm. 11, pp. 1291-1295
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The mechanism of allosteric coupling in choline kinase α1 revealed by the action of a rationally designed inhibitor
Angewandte Chemie - International Edition, Vol. 52, Núm. 17, pp. 4582-4586
2012
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1H and 13C NMR spectral assignments of pyridinium salts linked to a N-9 or N-3 adenine moiety
Magnetic Resonance in Chemistry, Vol. 50, Núm. 6, pp. 466-469
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Design, synthesis, theoretical calculations and biological evaluation of new non-symmetrical choline kinase inhibitors
European Journal of Medicinal Chemistry, Vol. 50, pp. 154-162
2007
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QSAR as a tool for the development of potent antiproliferative agents by inhibition of choline kinase
Current Computer-Aided Drug Design, Vol. 3, Núm. 4, pp. 297-313
2006
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(Q)SAR studies to design new human choline kinase inhibitors as antiproliferative drugs
Current Medicinal Chemistry, Vol. 13, Núm. 11, pp. 1231-1248
2005
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1H and 13C spectral assignment of symmetrical bis[(4-aminosubstituted)quinolinium] derivatives
Magnetic Resonance in Chemistry, Vol. 43, Núm. 12, pp. 1066-1071
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Symmetrical bis-quinolinium compounds: New human choline kinase inhibitors with antiproliferative activity against the HT-29 cell line
Journal of Medicinal Chemistry, Vol. 48, Núm. 9, pp. 3354-3363
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Towards a model for the inhibition of choline kinase by a new type of inhibitor
European Journal of Medicinal Chemistry, Vol. 40, Núm. 3, pp. 315-319