ANA
CONEJO GARCÍA
CATEDRÁTICA DE UNIVERSIDAD
ANTONIO
ENTRENA GUADIX
Investigador en el periodo 2009-2018
Publicaciones en las que colabora con ANTONIO ENTRENA GUADIX (15)
2017
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Choline kinase inhibition and docking studies of a series of 6-(benzylthio)-9H-purin-9-yl-pyridinium derivatives
Medicinal Chemistry Research, Vol. 26, Núm. 11, pp. 2809-2815
2016
2014
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Discovery of a new binding site on human choline kinase α1: Design, synthesis, crystallographic studies, and biological evaluation of asymmetrical bispyridinium derivatives
Journal of Medicinal Chemistry, Vol. 57, Núm. 2, pp. 507-515
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In vitro antiplasmodial and cytotoxic activities of asymmetrical pyridinium derivatives
European Journal of Medicinal Chemistry, Vol. 85, pp. 289-292
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NMR spectroscopic characterization of new nonsymmetrical bispyridinium choline kinase inhibitors
Magnetic Resonance in Chemistry
2013
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Antiproliferative activity, cell cycle, and apoptosis studies of a series of 6-substituted 9H-purin-9-yl-pyridinium derivatives on a human cervical carcinoma cell line
ChemMedChem, Vol. 8, Núm. 8, pp. 1266-1269
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Determination of potential scaffolds for human choline kinase α1 by chemical deconvolution studies
ChemBioChem, Vol. 14, Núm. 11, pp. 1291-1295
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The mechanism of allosteric coupling in choline kinase α1 revealed by the action of a rationally designed inhibitor
Angewandte Chemie - International Edition, Vol. 52, Núm. 17, pp. 4582-4586
2012
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1H and 13C NMR spectral assignments of pyridinium salts linked to a N-9 or N-3 adenine moiety
Magnetic Resonance in Chemistry, Vol. 50, Núm. 6, pp. 466-469
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Design, synthesis, theoretical calculations and biological evaluation of new non-symmetrical choline kinase inhibitors
European Journal of Medicinal Chemistry, Vol. 50, pp. 154-162
2007
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Cyclophanes and bicyclophanes: Fascinating molecules in organic chemistry
Targets in Heterocyclic Systems, Vol. 11, pp. 431-448
2006
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(Q)SAR studies to design new human choline kinase inhibitors as antiproliferative drugs
Current Medicinal Chemistry, Vol. 13, Núm. 11, pp. 1231-1248
2005
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Synthesis and NMR studies on a C3-symmetrical triquinolina triscationic bicyclophane
Journal of Organic Chemistry, Vol. 70, Núm. 14, pp. 5748-5751
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Towards a model for the inhibition of choline kinase by a new type of inhibitor
European Journal of Medicinal Chemistry, Vol. 40, Núm. 3, pp. 315-319
2003
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Conformational Dynamics of a Bispyridinium Cyclophane
Journal of Organic Chemistry, Vol. 68, Núm. 22, pp. 8697-8699