ANTONIO
ENTRENA GUADIX
Investigador en el periodo 2009-2018
Universidad de Zaragoza
Zaragoza, EspañaPublicaciones en colaboración con investigadores/as de Universidad de Zaragoza (7)
2017
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Choline kinase inhibition and docking studies of a series of 6-(benzylthio)-9H-purin-9-yl-pyridinium derivatives
Medicinal Chemistry Research, Vol. 26, Núm. 11, pp. 2809-2815
2016
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Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1)
Scientific Reports, Vol. 6
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Plasmodium falciparum Choline Kinase Inhibition Leads to a Major Decrease in Phosphatidylethanolamine Causing Parasite Death
Scientific Reports, Vol. 6
2015
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Pharmacophore-Based Virtual Screening to Discover New Active Compounds for Human Choline Kinase α1
Molecular Informatics, Vol. 34, Núm. 6-7, pp. 458-466
2014
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Choline kinase active site provides features for designing versatile inhibitors
Current Topics in Medicinal Chemistry, Vol. 14, Núm. 23, pp. 2684-2693
2013
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Determination of potential scaffolds for human choline kinase α1 by chemical deconvolution studies
ChemBioChem, Vol. 14, Núm. 11, pp. 1291-1295
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The mechanism of allosteric coupling in choline kinase α1 revealed by the action of a rationally designed inhibitor
Angewandte Chemie - International Edition, Vol. 52, Núm. 17, pp. 4582-4586