MARÍA DORA
CARRIÓN PEREGRINA
PROFESORA TITULAR DE UNIVERSIDAD
University of Ferrara
Ferrara, ItaliaPublicaciones en colaboración con investigadores/as de University of Ferrara (36)
2014
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Synthesis and biological evaluation of novel 2-amino-3-aroyl-4-neopentyl-5- substituted thiophene derivatives as allosteric enhancers of the A1 adenosine receptor
Bioorganic and Medicinal Chemistry, Vol. 22, Núm. 1, pp. 148-166
2013
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Synthesis and biological effects of novel 2-amino-3-(4-chlorobenzoyl)-4- substituted thiophenes as allosteric enhancers of the A1 adenosine receptor
European Journal of Medicinal Chemistry, Vol. 67, pp. 409-427
2012
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Structure-activity relationships of 2-amino-3-aroyl-4-[(4-arylpiperazin-1- yl)methyl]thiophenes. Part 2: Probing the influence of diverse substituents at the phenyl of the arylpiperazine moiety on allosteric enhancer activity at the A 1 adenosine receptor
Bioorganic and Medicinal Chemistry, Vol. 20, Núm. 2, pp. 996-1007
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Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[(4- arylpiperazin-1-yl)methyl]-5-substituted-thiophenes. Effect of the 5-modification on allosteric enhancer activity at the A1 adenosine receptor
Journal of Medicinal Chemistry, Vol. 55, Núm. 17, pp. 7719-7735
2011
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Synthesis and Antitumor Molecular Mechanism of Agents Based on Amino 2-(3',4',5'-Trimethoxybenzoyl)benzo[b]furan: Inhibition of Tubulin and Induction of Apoptosis
ChemMedChem, Vol. 6, Núm. 10, pp. 1841-1853
2010
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Substituted 2-(3′,4′,5′-trimethoxybenzoyl)-benzo[b] thiophene derivatives as potent tubulin polymerization inhibitors
Bioorganic and Medicinal Chemistry, Vol. 18, Núm. 14, pp. 5114-5122
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Symmetrical α-bromoacryloylamido diaryldienone derivatives as a novel series of antiproliferative agents. Design, synthesis and biological evaluation
Bioorganic and Medicinal Chemistry Letters, Vol. 20, Núm. 9, pp. 2733-2739
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Synthesis and antitumor activity of 1,5-disubstituted 1,2,4-triazoles as cis-restricted combretastatin analogues
Journal of Medicinal Chemistry, Vol. 53, Núm. 10, pp. 4248-4258
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Synthesis and evaluation of haloacetyl, α-bromoacryloyl and nitrooxyacetyl benzo[b]furan and benzo[b]thiophene derivatives as potent antiproliferative agents against leukemia l1210 and K562 cells
Letters in Drug Design and Discovery, Vol. 7, Núm. 7, pp. 476-486
2009
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2-Arylamino-4-amino-5-aroylthiazoles. "One-pot" synthesis and biological evaluation of a new class of inhibitors of tubulin polymerization
Journal of Medicinal Chemistry, Vol. 52, Núm. 17, pp. 5551-5555
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Design, synthesis and structure-activity relationship of 2-(3′,4′,5′-trimethoxybenzoyl)-benzo[b]furan derivatives as a novel class of inhibitors of tubulin polymerization
Bioorganic and Medicinal Chemistry, Vol. 17, Núm. 19, pp. 6862-6871
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Discovery of 8-methoxypyrazino[1,2-a]indole as a new potent antiproliferative agent against human leukemia K562 cells. A structure-activity relationship study
Letters in Drug Design and Discovery, Vol. 6, Núm. 4, pp. 298-303
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Hybrid α-bromoacryloylamido chalcones. Design, synthesis and biological evaluation
Bioorganic and Medicinal Chemistry Letters, Vol. 19, Núm. 7, pp. 2022-2028
2008
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Design, synthesis, and biological evaluation of thiophene analogues of chalcones
Bioorganic and Medicinal Chemistry, Vol. 16, Núm. 10, pp. 5367-5376
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Synthesis and biological evaluation of 1-methyl-2-(3′,4′, 5′-trimethoxybenzoyl)-3-aminoindoles as a new class of antimitotic agents and tubulin inhibitors
Journal of Medicinal Chemistry, Vol. 51, Núm. 5, pp. 1464-1468
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Synthesis and biological evaluation of 2-(3′,4′,5′-trimethoxybenzoyl)-3-N,N-dimethylamino benzo[b]furan derivatives as inhibitors of tubulin polymerization
Bioorganic and Medicinal Chemistry, Vol. 16, Núm. 18, pp. 8419-8426
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Synthesis and biological evaluation of 2-amino-3-(3′,4′,5′-trimethoxybenzoyl)-6-substituted-4 ,5,6,7-tetrahydrothieno[2,3-c]pyridine derivatives as antimitotic agents and inhibitors of tubulin polymerization
Bioorganic and Medicinal Chemistry Letters, Vol. 18, Núm. 18, pp. 5041-5045
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Synthesis and biological evaluation of 2-amino-3-(4-chlorobenzoyl)-4-[N- (substituted) piperazin-1-yl]thiophenes as potent allosteric enhancers of the A1 adenosine receptor
Journal of Medicinal Chemistry, Vol. 51, Núm. 18, pp. 5875-5879
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Synthesis and biological evaluation of 2-aroyl-4-phenyl-5-hydroxybenzofurans as a new class of antitubulin agents
Medicinal Chemistry, Vol. 4, Núm. 6, pp. 558-564
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Synthesis and biological evaluation of a series of 2-(3,4,5- trimethoxybenzoyl)-indol-3-yl acetic acid derivatives as potential agents against human leukemia K562 cells
Letters in Drug Design and Discovery, Vol. 5, Núm. 3, pp. 214-220