ANTONIO
ENTRENA GUADIX
Investigador en el periodo 2009-2018
MIGUEL ÁNGEL
GALLO MEZO
Investigador en el periodo 2002-2017
Publicaciones en las que colabora con MIGUEL ÁNGEL GALLO MEZO (63)
2018
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Lead optimization-hit expansion of new asymmetrical pyridinium/quinolinium compounds as choline kinase α1 inhibitors
Future Medicinal Chemistry, Vol. 10, Núm. 15, pp. 1769-1786
2016
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1H and 13C NMR spectral assignments of 1,1′-(((ethane-1,2-diylbis(oxy))bis(4,1-phenylene))bis(methylene))-bispyridinium and -bisquinolinium bromide derivatives
Magnetic Resonance in Chemistry
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Design, synthesis, crystallization and biological evaluation of new symmetrical biscationic compounds as selective inhibitors of human Choline Kinase α1 (ChoKα1)
Scientific Reports, Vol. 6
2015
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New more polar symmetrical bipyridinic compounds: New strategy for the inhibition of choline kinase α1
Future Medicinal Chemistry, Vol. 7, Núm. 4, pp. 417-436
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New more polar symmetrical choline kinase inhibitors II: Study of setting up a new scaffold for the cancer therapy
Journal of Biological Research (Italy)
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Pharmacophore-Based Virtual Screening to Discover New Active Compounds for Human Choline Kinase α1
Molecular Informatics, Vol. 34, Núm. 6-7, pp. 458-466
2014
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1H, 13C NMR studies of new 3-aminophenol isomers linked to pyridinium salts
Magnetic Resonance in Chemistry, Vol. 52, Núm. 1-2, pp. 40-46
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Discovery of a new binding site on human choline kinase α1: Design, synthesis, crystallographic studies, and biological evaluation of asymmetrical bispyridinium derivatives
Journal of Medicinal Chemistry, Vol. 57, Núm. 2, pp. 507-515
2013
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Antiproliferative activity, cell cycle, and apoptosis studies of a series of 6-substituted 9H-purin-9-yl-pyridinium derivatives on a human cervical carcinoma cell line
ChemMedChem, Vol. 8, Núm. 8, pp. 1266-1269
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New non-symmetrical choline kinase inhibitors
Bioorganic and Medicinal Chemistry, Vol. 21, Núm. 22, pp. 7146-7154
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Synthesis and biological evaluation of 4,5-dihydro-1H-pyrazole derivatives as potential nNOS/iNOS selective inhibitors. Part 2: Influence of diverse substituents in both the phenyl moiety and the acyl group
Bioorganic and Medicinal Chemistry, Vol. 21, Núm. 14, pp. 4132-4142
2012
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1H and 13C NMR spectral assignments of pyridinium salts linked to a N-9 or N-3 adenine moiety
Magnetic Resonance in Chemistry, Vol. 50, Núm. 6, pp. 466-469
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1,3,4-Thiadiazole derivatives as selective inhibitors of iNOS versus nNOS: Synthesis and structure-activity dependence
European Journal of Medicinal Chemistry, Vol. 50, pp. 129-139
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Characterization of 4,5-Dihydro-1H-Pyrazole Derivatives by 13C NMR Spectroscopy
Magnetic Resonance in Chemistry, Vol. 50, Núm. 1, pp. 58-61
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Design, synthesis, theoretical calculations and biological evaluation of new non-symmetrical choline kinase inhibitors
European Journal of Medicinal Chemistry, Vol. 50, pp. 154-162
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Melatonin synthetic analogs as nitric oxide synthase inhibitors
Mini-Reviews in Medicinal Chemistry, Vol. 12, Núm. 7, pp. 600-617
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NMR spectroscopic characterization of new 2,3-dihydro-1,3,4-thiadiazole derivatives
Magnetic Resonance in Chemistry, Vol. 50, Núm. 7, pp. 515-522
2011
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Utilización y aplicación de la herramienta "google docs" en la docencia universitaria dentro del marco del EEES
Univest 2011: III Congreso Internacional "La autogestión del aprendizaje" (Universitat de Girona = Universidad de Gerona)
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Utilización y aplicación de la herramienta "google docs" en la docencia universitaria dentro del marco del EEES
, pp. 51
2009
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Melatonin and its brain metabolite N1-acetyl-5-methoxykynuramine prevent mitochondrial nitric oxide synthase induction in Parkinsonian mice
Journal of Neuroscience Research, Vol. 87, Núm. 13, pp. 3002-3010